An Efficient Synthesis of Arylated Pyridines from Conjugated Acetylenes and Substituted Benzylamines Catalyzed by Base.
نویسندگان
چکیده
An efficient base-catalyzed synthesis of arylated pyridines has been disclosed. This reaction involving conjugated acetylenes and substituted benzylamines proceeded smoothly, giving rise to tri-aryl substituted pyridines which are biologically relevant compounds in good to excellent yields in N,N-dimethylformamide (DMF) under air at 140 °C with K₂CO₃ as catalyst.
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ورودعنوان ژورنال:
- Molecules
دوره 22 8 شماره
صفحات -
تاریخ انتشار 2017